Category: 152626-77-2

On September 15, 2022, Baugh, Simon David Peter; Freeman, Kathryn B.; Pelletier, Jeffrey Claude; Reitz, Allen B.; Scott, Richard W.; Weaver, Damian G.; Whitman, David B. published a patent.Application of 152626-77-2 The title of the patent was Novel heteroaromatic compounds exhibiting antifungal activity and their method of use and preparation. And the patent contained the following:

Pharmaceutical compositions of the invention comprise heteroaromatic compounds of formula I having a disease-modifying action in the treatment of fungal infections and diseases associated with fungal infection. Compounds of formula I wherein A1 is (un)substituted thiazolyl, (un)substituted thiadiazolyl, (un)substituted imidazolyl, (un)substituted pyrazinyl, etc.; A2 is (un)substituted pyrimidinyl, (un)substiuted pyrazinyl, (un)substituted oxadiazolyl, (un)substituted thiadiazolyl, etc.; A3 is (CH2)0-2NHC:NHNH2 and derivatives, (CH2)0-2C:NHNH2 and derivatives, OCH2CH2NHC:NHNH2 and derivatives, etc.; A4 is (CH2)0-3NHC:NHNH2 and derivatives, (CH2)0-3C:NHNH2 and derivatives, OCH2CH2NHC:NHNH2 and derivatives, etc.; R1 is H, C1-4 alkyl and C3-5 branched alkyl; and enantiomers, diastereomers, hydrates, solvates, pharmaceutically acceptable salts, prodrugs and complexes thereof, are claimed. Example compound II•2TFA was prepared by a multistep procedure (procedure given). The invention compound were evaluated for their antifungal activity (data given). The experimental process involved the reaction of 4-Bromo-5-methoxy-2-methylaniline(cas: 152626-77-2).Application of 152626-77-2

The Article related to heteroaromatic preparation antifungal, Heterocyclic Compounds (More Than One Hetero Atom): Pyrazines and Quinoxalines (Including Piperazines) and other aspects.Application of 152626-77-2

Referemce:
Ether – Wikipedia,
Ether | (C2H5)2O – PubChem

On September 16, 1993, James, Donald R.; Baker, Don R.; Mielich, Steven D.; Michaely, William J.; Fitzjohn, Steven; Knudsen, Christopher G.; Mathews, Christopher; Gerdes, John M. published a patent.Category: ethers-buliding-blocks The title of the patent was Preparation of arylindazoles and their use as herbicides. And the patent contained the following:

Title compounds I (R1 = H, halo; R2 = H, O2N, halo, alkyl, NC, alkylthio, alkylsulfinyl, alkylsulfonyl, alkoxy, AcNH, H2N; R3 = H, halo, haloalkyl, haloalkoxy, NC, H2N, R13OyS wherein R13 = alkyl, haloalkyl, y = 0-2; R4, R5, R6 = H, halo, O2N, HO, NC, alkyl, alkoximinoalkyl, hydroxyalkyl, haloalkyl, CHO, etc.; R7 = H, halo, alkyl, O2N; R8 = H, halo; X = N, R14C wherein R14 = H, halo, haloalkyl, NC, etc.) and salts thereof, are prepared 6-Imidazolol in DMF was reacted with K2CO3 followed by MeI to give 6-methoxyindazole which in DMF was treated with 3,5,4-Cl2FC6H2CF3 and K2CO3 to give I (R1 = R4 = R5 = R7 = R8 = H, R2 = Cl, R3 = F3C, R6 = MeO, X = ClC) (II) in preemergence application II at 4 kg/ha showed 100% herbicidal effect against green foxtail, watergrass, wild mustard, velvetleaf, etc. A large number of I were prepared and evaluated both pre- and postemergence. The experimental process involved the reaction of 4-Bromo-5-methoxy-2-methylaniline(cas: 152626-77-2).Category: ethers-buliding-blocks

The Article related to indazole aryl preparation herbicide, Heterocyclic Compounds (More Than One Hetero Atom): Other 5-Membered Rings, Two Or More Hetero Atoms and other aspects.Category: ethers-buliding-blocks

Referemce:
Ether – Wikipedia,
Ether | (C2H5)2O – PubChem

On May 24, 2018, Weiss, Matthias; Sulzer-Mosse, Sarah published a patent.Related Products of 152626-77-2 The title of the patent was Preparation of microbiocidal phenylamidine derivatives. And the patent contained the following:

Compounds of the formula I, wherein R1 and R2 are independently C1-4 alkyl and C3-6 cycloalkyl; R3 is H, halo, C1-4 alkyl, etc.; R4 is haloalkyl; R5 is C3-8 (un)substituted cycloalkyl, C1-6 alkyloxycarbonyl, (un)substituted C1-6 alkyl. Furthermore, the invention relates to agrochem. compositions which comprise compounds of formula I, to preparation of these compositions, and to the use of the compounds or compositions in agriculture or horticulture for combating, preventing or controlling infestation of plants, harvested food crops, seeds or non-living materials by phytopathogenic microorganisms, in particular fungi. Example compound II was prepared by a multistep procedure starting with 5-methoxy-2-methylaniline. The experimental process involved the reaction of 4-Bromo-5-methoxy-2-methylaniline(cas: 152626-77-2).Related Products of 152626-77-2

The Article related to phenylamidine preparation microbiocidal agriculture horticulture, Benzene, Its Derivatives, and Condensed Benzenoid Compounds: Amides, Amidines, Imidic Esters, Hydrazides, and Hydrazonic Esters and other aspects.Related Products of 152626-77-2

Referemce:
Ether – Wikipedia,
Ether | (C2H5)2O – PubChem

On December 20, 2018, Weiss, Matthias; Sulzer-Mosse, Sarah published a patent.Category: ethers-buliding-blocks The title of the patent was N-phenyl amidine derivatives used in fungicidal compositions and their preparation. And the patent contained the following:

The invention relates compounds of formula I and their use as fungicides. Compounds of formula I, wherein R1 is Et, isopropy and cyclopropyl, R2 is cyclopropyl, n-butoxymethyl, Ph, etc.; and salts, enantiomers, tautomers and N-oxides thereof, are claimed. Compound II was prepared by halogenation of 5-methoxy-2-methyl-aniline with N-bromosuccinimide to give 4-bromo-5-methoxy-2-methyl-aniline, the resulting compound underwent N-alkylation with N-(dimethoxymethyl)-N-methyl-ethanamine which resulted in compound II. Compounds of the invention were tested for their fungicidal activity (data given). The experimental process involved the reaction of 4-Bromo-5-methoxy-2-methylaniline(cas: 152626-77-2).Category: ethers-buliding-blocks

The Article related to phenyl amidine preparation fungicide phytopathogenic, Benzene, Its Derivatives, and Condensed Benzenoid Compounds: Amides, Amidines, Imidic Esters, Hydrazides, and Hydrazonic Esters and other aspects.Category: ethers-buliding-blocks

Referemce:
Ether – Wikipedia,
Ether | (C2H5)2O – PubChem